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Naslov Design of fluorinated triazinoindoles as highly potent and markedly selective ALR2 inhibitors: synthesis, in silico and in vitro evaluation of promising lead compounds (Article)
Autori Kovacikova Lucia  Teplanova Terezia  Majekova Magdalena  Almassy Ambroz  Addova Gabriela  Hanquet Gilles  Pannosian Armen  Dobricic Vladimir  Savic Jelena  Bohac Andrej 
Info BIOORGANIC CHEMISTRY, (2026), vol. 181 br. , str. -
Projekat Slovak Grant Agency [VEGA 2/0124/26, VEGA 2/0136/26]; Slovak Research and Development Agency [APVV-24-0388, APVV DS-FR-24-0052]; Ministry of Science, Technological Development, and Innovation of the Republic of Serbia [451-03-33/2026-03/200161, 451-03-34/2026-03/200161]
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Naslov Selectivity of N(2)-substituted oxotriazinoindole aldose reductase inhibitors is determined by the interaction pattern with Pro301-Arg312 loop of aldehyde reductase (Article)
Autori Kovacikova Lucia  Gaikwad Sunil  Almasiova Kristina  Almassy Ambroz  Addova Gabriela  Majekova Magdalena  Hanquet Gilles  Dobricic Vladimir D  Bohac Andrej  Stefek Milan 
Info MEDICINAL CHEMISTRY RESEARCH, (2024), vol. 33 br. 3, str. 492-503
Projekat Vedeck Grantov Agentra MScaron;VVaScaron; SR a SAV [2/0008/22, VEGA 2/0103/22, APVV-20-0411, APVV-20-0543, APVV SK-SRB-21-0047 (451-03-43/2022-09/02)]; VEGA; Ministry of Science, Technological Development and Innovation, Republic of Serbia [SK-FR-22-0017]; University of Belgrade-Faculty of Pharmacy, APVV [ITMS2014+: 313021x329, ITMS2014+: 313021BUZ3]; Advancing University Capacity and Competence in Research, Development and Innovation (Accord); European Regional Development Fund
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